SCHEMBL3955015

SCHEMBL3955015

COc1cc(Cl)c(-c2nc(SCC(=O)NC3CC3)nc3c2c(C#N)cn3COCC[Si](C)(C)C)cc1O

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 8/20 0.53
HSP90AA1 P07900 3/20 0.52
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
KCNH2 Q12809 3/20 0.39
LMNA P02545 2/20 0.37
RXFP1 Q9HBX9 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
KMT2A Q03164 2/20 0.34
RAB9A P51151 1/20 0.34
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3961248 0.91 HSP90AB1 (0.56) HSP90AB1HSP90AA1KCNH2LMNARXFP1
SCHEMBL3961239 0.87 HSP90AA1 (0.56) HSP90AB1HSP90AA1GAAKCNH2
SCHEMBL4134884 0.86 HSP90AB1 (0.50) HSP90AB1HSP90AA1KDM4EALDH1A1MAPT
SCHEMBL3955021 0.84 HSP90AB1 (0.43) HSP90AB1HSP90AA1KCNH2
SCHEMBL4064357 0.83 HSP90AB1 (0.48) HSP90AB1HSP90AA1KCNH2TDP1KMT2A
SCHEMBL2569133 0.82 HSP90AB1 (0.46) HSP90AB1HSP90AA1KCNH2
SCHEMBL3961415 0.82 HSP90AB1 (0.51) HSP90AB1HSP90AA1KCNH2LMNA
SCHEMBL3955735 0.82 HSP90AA1 (0.62) HSP90AB1HSP90AA1KCNH2
SCHEMBL3956211 0.81 HSP90AB1 (0.47) HSP90AB1HSP90AA1KDM4EALDH1A1GAA
SCHEMBL4059825 0.81 HSP90AB1 (0.45) HSP90AB1HSP90AA1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009030871-A1 PYRROLOPYRIMIDINE DERIVATIVES HAVING HSP90 INHIBITORY ACTIVITY VERNALIS R & D LTD (GB) 2009-03-12 WO disclosed