SCHEMBL3958415

SCHEMBL3958415

C[C@H](NC(=O)O)[C@@H](N)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 4/20 0.40
ALDH1A1 P00352 1/20 0.40
TACR1 P25103 8/20 0.40
MAPT P10636 1/20 0.38
CES2 O00748 1/20 0.38
CYP2D6 P10635 2/20 0.38
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
TACR3 P29371 1/20 0.38
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3958410 1.00 SCN9A (0.40) SCN9AALDH1A1TACR1MAPTCES2
SCHEMBL15062085 0.84 ALDH1A1 (0.42) ALDH1A1TACR1MAPTCES2CYP2D6
SCHEMBL4234698 0.83 ALDH1A1 (0.41) ALDH1A1TACR1MAPTCES2CYP2D6
SCHEMBL3950662 0.83 ALDH1A1 (0.41) ALDH1A1TACR1MAPTCES2CYP2D6
SCHEMBL4234694 0.83 ALDH1A1 (0.41) ALDH1A1TACR1MAPTCES2CYP2D6
SCHEMBL15821803 0.83 ALDH1A1 (0.41) ALDH1A1TACR1MAPTCES2CYP2D6
SCHEMBL3950088 0.81 SCN9A (0.40) SCN9AALDH1A1TACR1MAPTCES2
SCHEMBL17200949 0.81 CES2 (0.42) ALDH1A1TACR1MAPTCES2CYP2D6
SCHEMBL13905599 0.77 TACR1 (0.48) SCN9AALDH1A1TACR1
SCHEMBL18989371 0.75 CXCR2 (0.38) SCN9AALDH1A1TACR1PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009027785-A2 1, 3-OXAZOLE DERIVATIVES AS CETP INHIBITORS PFIZER PRODUCTS INC. (US) 2009-03-05 WO disclosed