SCHEMBL3958441

SCHEMBL3958441

CCc1cnc(C)cn1.NN=O

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.33
NOS2 P35228 2/20 0.33
NOS1 P29475 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
CYP1A2 P05177 4/20 0.31
CYP3A4 P08684 4/20 0.31
CLK4 Q9HAZ1 3/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
POLB P06746 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL110053 0.87
Formamide SCHEMBL28177237 0.84 NOS3 (0.33) NOS3NOS2NOS1L3MBTL1CYP1A2
Pyrrole SCHEMBL25253437 0.76 CYP1A2 (0.33) CYP1A2CYP3A4CLK4MEN1KMT2A
SCHEMBL830188 0.75 NOS3 (0.33) NOS3NOS2NOS1CYP1A2POLB
SCHEMBL28249551 0.74 CYP3A4 (0.37) CYP1A2CYP3A4CLK4MEN1KMT2A
SCHEMBL29411708 0.73 CYP3A4 (0.33) CYP1A2CYP3A4CLK4MEN1KMT2A
Valine SCHEMBL16597282 0.73 SLC7A5 (0.46) L3MBTL1POLB
SCHEMBL29412844 0.72
SCHEMBL5476 0.72
SCHEMBL27778974 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079756-A2 SYNTHETIC PEPTIDE AMIDES AND DIMERS THEREOF Cara Therapeutics, Inc. (US) 2009-07-22 EP disclosed
WO-2008060552-A2 SYNTHETIC PEPTIDE AMIDES AND DIMERS THEREOF CARA THERAPEUTICS, INC. (US) 2008-05-22 WO disclosed