SCHEMBL3961313

SCHEMBL3961313

O=C(O)N1CCC(O)(CS)CC1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 1/20 0.32
ALDH1A1 P00352 2/20 0.31
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4076810 0.92
SCHEMBL23253117 0.80 CYP46A1 (0.33) AVPR1AALDH1A1LMNAGAASMN1; SMN2
SCHEMBL1972942 0.78 SLC6A2 (0.33) AVPR1AALDH1A1LMNAGAASMN1; SMN2
SCHEMBL21840110 0.78 CYP46A1 (0.40) AVPR1AALDH1A1LMNAGAASMN1; SMN2
SCHEMBL20702372 0.78 AVPR1A (0.32) AVPR1AALDH1A1LMNAGAASMN1; SMN2
SCHEMBL238639 0.77 PKLR (0.34) AVPR1AALDH1A1LMNA
SCHEMBL28219846 0.75 CYP2D6 (0.32) AVPR1AALDH1A1LMNA
SCHEMBL2141413 0.75 AVPR1A (0.31) AVPR1AALDH1A1LMNA
SCHEMBL10694845 0.75 L3MBTL1 (0.51) ALDH1A1LMNAGAASMN1; SMN2
SCHEMBL4765795 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035435-A1 NOVEL LAPACHONE COMPOUNDS AND METHODS OF USE THEREOF ARQULE, INC. (US) 2009-03-18 EP disclosed
WO-2007139569-A1 NOVEL LAPACHONE COMPOUNDS AND METHODS OF USE THEREOF ARQULE, INC. (US) 2007-12-06 WO disclosed