SCHEMBL3961835

SCHEMBL3961835

CC(C)(C)OC(=O)N[C@H](C(=O)O)C1CC2CCC(C1)N2C(=O)c1ncccc1F

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.38
SCN9A Q15858 5/20 0.37
CYP3A4 P08684 4/20 0.37
HCRTR1 O43613 3/20 0.37
HCRTR2 O43614 3/20 0.37
MMP13 P45452 2/20 0.37
SCN10A Q9Y5Y9 3/20 0.36
GPR119 Q8TDV5 3/20 0.36
JAK2 O60674 2/20 0.35
JAK1 P23458 2/20 0.35
METAP1 P53582 1/20 0.35
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
PTPN1 P18031 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3751314 0.87 MMP13 (0.37) AAK1SCN9ACYP3A4HCRTR1HCRTR2
SCHEMBL3753926 0.83 MMP13 (0.42) AAK1MMP13GPR119JAK2JAK1
SCHEMBL3738226 0.81 MGLL (0.39) AAK1MMP13GPR119JAK2JAK1
SCHEMBL3736510 0.81 MGLL (0.39) AAK1MMP13GPR119JAK2JAK1
SCHEMBL3738694 0.81 PREP (0.38) AAK1HCRTR1HCRTR2MMP13GPR119
SCHEMBL3745735 0.81 BCL2 (0.45) CYP3A4
SCHEMBL3751575 0.80 MMP13 (0.41) AAK1MMP13JAK2JAK1
SCHEMBL3741700 0.79 AAK1 (0.40) AAK1MMP13
SCHEMBL3747163 0.79 AAK1 (0.41) AAK1SCN9AHCRTR1HCRTR2MMP13
SCHEMBL3742665 0.78 KDM4D (0.36) AAK1CYP3A4MMP13GPR119JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009037719-A1 NOVEL COMPOUNDS AS DIPEPTIDYL PEPTIDASE IV (DPP IV) INHIBITORS LUPIN LIMITED (IN) 2009-03-26 WO disclosed