SCHEMBL3961945

SCHEMBL3961945

COC(=O)c1ccncc1CC(C)C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.55
KDM4E B2RXH2 4/20 0.55
GLA P06280 1/20 0.55
GAA P10253 1/20 0.55
KDM4C Q9H3R0 4/20 0.46
KDM6B O15054 1/20 0.46
LMNA P02545 3/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CDK4 P11802 1/20 0.42
CCND1 P24385 1/20 0.42
GSK3B P49841 1/20 0.42
MAPK8 P45983 1/20 0.41
MAPK9 P45984 1/20 0.41
MAPK10 P53779 1/20 0.41
KMT2A Q03164 2/20 0.40
HSD17B10 Q99714 2/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
CYP46A1 Q9Y6A2 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845125 0.87 ALDH1A1 (0.62) ALDH1A1KDM4EGLAGAAKDM4C
SCHEMBL25827431 0.84 ALDH1A1 (0.58) ALDH1A1KDM4EGLAGAAKDM4C
SCHEMBL28613135 0.82 ALDH1A1 (0.60) ALDH1A1KDM4EGLAGAAKDM4C
SCHEMBL23639428 0.81 ALDH1A1 (0.58) ALDH1A1KDM4EGLAGAAKDM4C
SCHEMBL21786269 0.81 ALDH1A1 (0.63) ALDH1A1KDM4EGLAGAAKDM4C
SCHEMBL15832960 0.79 ALDH1A1 (0.57) ALDH1A1KDM4EGLAGAAKDM4C
SCHEMBL29323004 0.79 ALDH1A1 (0.47) ALDH1A1KDM4EGLAGAAKDM4C
SCHEMBL19838578 0.77 ALDH1A1 (0.54) ALDH1A1KDM4EGLAGAAKDM4C
SCHEMBL23674679 0.77 ALDH1A1 (0.54) ALDH1A1KDM4EGLAGAAKDM4C
SCHEMBL29792765 0.77 ALDH1A1 (0.54) ALDH1A1KDM4EGLAGAAKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-A2 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2009-07-22 EP disclosed
WO-2008038251-A2 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-04-03 WO disclosed