SCHEMBL3962265

SCHEMBL3962265

O=C1Nc2cc(Cl)ccc2C1(Cc1cccc(Cl)c1)C1CCCNC1

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 11/20 0.64
TP53 P04637 10/20 0.64
SSTR1 P30872 1/20 0.39
SSTR4 P31391 1/20 0.39
DRD2 P14416 1/20 0.37
MAOB P27338 1/20 0.37
PKM P14618 1/20 0.36
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3969681 0.88 MDM2 (0.69) MDM2TP53MAOB
SCHEMBL3962743 0.87 MDM2 (0.62) MDM2TP53SSTR1SSTR4MAOB
SCHEMBL3966408 0.83 MDM2 (0.64) MDM2TP53MAOB
SCHEMBL3966209 0.82 MDM2 (0.62) MDM2TP53SSTR1SSTR4MAOB
SCHEMBL3964393 0.81 MDM2 (0.60) MDM2TP53PKM
SCHEMBL4962890 0.79 MDM2 (0.77) MDM2TP53
SCHEMBL3969547 0.79 MDM2 (0.71) MDM2TP53DRD2
SCHEMBL3964720 0.79 MDM2 (0.86) MDM2TP53
SCHEMBL4966721 0.78 MDM2 (0.70) MDM2TP53
SCHEMBL19571070 0.78 MDM2 (0.52) MDM2TP53SSTR1SSTR4MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7576082-B2 Oxindole derivatives HOFFMAN-LA ROCHE INC. (US) 2009-08-18 US disclosed
US-7576082-B2 Oxindole derivatives HOFFMAN-LA ROCHE INC. (US) 2009-08-18 US disclosed
US-7576082-B2 Oxindole derivatives HOFFMAN-LA ROCHE INC. (US) 2009-08-18 US disclosed
EP-1896412-A2 OXINDOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2008-03-12 EP disclosed
WO-2006136606-A2 OXINDOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2006-12-28 WO disclosed
WO-2006136606-A2 OXINDOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2006-12-28 WO disclosed
US-20060293319-A1 Oxindole derivatives LUK KIM-CHUN 2006-12-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060293319-A1 Oxindole derivatives CCNI, OGFR, MKI67 MDM2 759/4885TP53 96/4885SSTR1 946/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.