SCHEMBL3963475

SCHEMBL3963475

COC(=O)Oc1cc(C)c2nc(C)[nH]c2c1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
DHODH Q02127 11/20 0.39
MME P08473 1/20 0.38
HTT P42858 1/20 0.37
PARP1 P09874 2/20 0.36
HSP90AA1 P07900 1/20 0.34
ESR2 Q92731 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3962137 0.85 DHODH (0.43) ALDH1A1HPGDDHODHMMEHTT
SCHEMBL4240634 0.81 MAPT (0.39) ALDH1A1
SCHEMBL3960529 0.81 PARP1 (0.42) HTTPARP1
SCHEMBL10288043 0.79 HTT (0.44) ALDH1A1DHODHHTTPARP1
SCHEMBL6170448 0.76 KDM4E (0.45) ALDH1A1HPGDDHODHMMEHTT
SCHEMBL6924904 0.74 DHODH (0.39) DHODHMMEHTTHSP90AA1ESR2
SCHEMBL6926116 0.74 SMN1; SMN2 (0.55) DHODHMME
SCHEMBL6502505 0.73 AR (0.43) ALDH1A1HPGDDHODHMMEHTT
SCHEMBL1542506 0.73 MAPT (0.37) ALDH1A1HPGDTDP1
SCHEMBL6923484 0.72 MCL1 (0.47) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034029-A2 1-SUBSTITUTED 4-HETEROCYCLYLPIPERIDINES FOR USE AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-19 WO disclosed