SCHEMBL3963655

SCHEMBL3963655

O=C(O)c1cc(F)c(F)nc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.53
NFE2L2 Q16236 1/20 0.53
KDM4E B2RXH2 3/20 0.44
ASPH Q12797 3/20 0.44
KDM8 Q8N371 2/20 0.44
NAPRT Q6XQN6 1/20 0.41
ALB P02768 2/20 0.38
AKR1C2 P52895 1/20 0.36
AKR1C1 Q04828 1/20 0.36
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ALDH1A1 P00352 3/20 0.33
ALOX15 P16050 2/20 0.33
ACMSD Q8TDX5 2/20 0.33
HIF1A Q16665 2/20 0.33
HCAR2 Q8TDS4 1/20 0.33
TSHR P16473 1/20 0.33
CYP1A2 P05177 1/20 0.33
AURKA O14965 1/20 0.33
DHODH Q02127 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7535033 0.83 KEAP1 (0.50) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL7591627 0.81 KEAP1 (0.48) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL19679344 0.81 KEAP1 (0.75) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL6837965 0.78 KDM4E (0.41) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL1300386 0.78 KEAP1 (0.41) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL8564557 0.77 KEAP1 (0.44) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL1301581 0.75 KEAP1 (0.39) KEAP1NFE2L2KDM4EASPHKDM8
SCHEMBL7858377 0.75 NPC1 (0.41) KDM4ENPC1RAB9AALDH1A1TSHR
SCHEMBL3960162 0.75 MAPT (0.41) KEAP1NFE2L2KDM4EALDH1A1CYP1A2
SCHEMBL4830274 0.75 KEAP1 (0.54) KEAP1NFE2L2KDM4EASPHKDM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014023531-A1 TRIFLUOROMETHYLPYRIDINE CARBOXAMIDES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2014-02-13 WO disclosed
EP-2079734-A1 OXADIAZOLE AND THIADIAZOLE COMPOUNDS AND THEIR USE AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS NeuroSearch A/S (DK) 2009-07-22 EP disclosed
WO-2008049864-A1 OXADIAZOLE AND THIADIAZOLE COMPOUNDS AND THEIR USE AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS NEUROSEARCH A/S (DK) 2008-05-02 WO disclosed