SCHEMBL3963945

SCHEMBL3963945

Cc1c(C(N)=O)cccc1-c1c[nH]c(=O)c(CNc2ccc(N3CCC(C)(O)CC3)nn2)c1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
STK4 Q13043 1/20 0.34
STK3 Q13188 1/20 0.34
PTGER4 P35408 2/20 0.31
PRKD1 Q15139 1/20 0.31
PRKD2 Q9BZL6 1/20 0.31
SCD O00767 1/20 0.31
JAK1 P23458 1/20 0.31
JAK3 P52333 1/20 0.31
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
CD38 P28907 1/20 0.30
KCNH2 Q12809 1/20 0.30
BDKRB1 P46663 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3965808 0.89 PIK3CB (0.37) STK4STK3PTGER4PRKD2JAK1
SCHEMBL4193391 0.88 AURKA (0.33) PRKD1PRKD2NPC1RAB9ACD38
SCHEMBL3740333 0.76 AURKA (0.39) PRKD1PRKD2NPC1RAB9A
SCHEMBL3744921 0.76 BTK (0.43) JAK1JAK3
SCHEMBL3750774 0.75 NPC1 (0.42) STK4STK3NPC1RAB9A
SCHEMBL3753112 0.73 ACVR1 (0.39) STK4STK3NPC1RAB9A
SCHEMBL3964701 0.69 BTK (0.45)
SCHEMBL3968942 0.66 BTK (0.51)
SCHEMBL3747925 0.65 BTK (0.42)
SCHEMBL3744929 0.65 BTK (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079726-A2 SUBSTITUTED AMIDES, METHOD OF MAKING, AND METHOD OF USE THEREOF CGI Pharmaceuticals, Inc. (US) 2009-07-22 EP disclosed
WO-2008033857-A2 SUBSTITUTED AMIDES, METHOD OF MAKING, AND METHOD OF USE THEREOF CGI PHARMACEUTICALS, INC. (US) 2008-03-20 WO disclosed