SCHEMBL4193391

SCHEMBL4193391

CCN1CCN(c2ccc(NCc3cc(-c4cccc(C(N)=O)c4C)c[nH]c3=O)nn2)CC1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.33
AURKB Q96GD4 2/20 0.33
BDKRB1 P46663 1/20 0.33
EZH1 Q92800 2/20 0.33
EZH2 Q15910 1/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
PARP1 P09874 4/20 0.32
PARP2 Q9UGN5 2/20 0.32
KIT P10721 1/20 0.32
PRKD1 Q15139 1/20 0.31
PRKD2 Q9BZL6 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
KDR P35968 1/20 0.31
MT-CO2 P00403 1/20 0.31
HRH4 Q9H3N8 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3965808 0.90 PIK3CB (0.37) AURKAAURKBNPC1RAB9APRKD2
SCHEMBL3963945 0.88 STK4 (0.34) BDKRB1NPC1RAB9APRKD1PRKD2
SCHEMBL3740333 0.78 AURKA (0.39) AURKAAURKBNPC1RAB9APARP1
SCHEMBL3757117 0.76 BTK (0.43)
SCHEMBL3750774 0.76 NPC1 (0.42) NPC1RAB9AKDM4E
SCHEMBL3753112 0.72 ACVR1 (0.39) NPC1RAB9APARP1
SCHEMBL3745143 0.67 BTK (0.41)
SCHEMBL3749975 0.67 BTK (0.41)
SCHEMBL3968942 0.66 BTK (0.51) AURKAAURKB
SCHEMBL3740338 0.66 AURKA (0.37) AURKAAURKBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079726-A2 SUBSTITUTED AMIDES, METHOD OF MAKING, AND METHOD OF USE THEREOF CGI Pharmaceuticals, Inc. (US) 2009-07-22 EP disclosed
WO-2008033857-A2 SUBSTITUTED AMIDES, METHOD OF MAKING, AND METHOD OF USE THEREOF CGI PHARMACEUTICALS, INC. (US) 2008-03-20 WO disclosed