SCHEMBL3964057

SCHEMBL3964057

COCCN(CCOC)C(=O)c1ccc(N(C)c2cc(-c3cccc(NC(=O)c4cc5c(s4)CCCC5)c3C)c[nH]c2=O)nc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.47
BTK Q06187 16/20 0.43
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3964067 0.89 BTK (0.44) BTKALDH1A1HPGDSMN1; SMN2KDM4E
SCHEMBL3956979 0.89 BTK (0.47) BTKALDH1A1HPGDSMN1; SMN2KDM4E
SCHEMBL3969273 0.88 BTK (0.46) BTKALDH1A1HPGDSMN1; SMN2KDM4E
SCHEMBL1323341 0.78 BTK (0.68) TDP1BTK
SCHEMBL1322896 0.78 BTK (0.67) TDP1BTK
SCHEMBL13893940 0.75 BTK (0.53) BTKALDH1A1HPGDSMN1; SMN2KDM4E
SCHEMBL1323039 0.74 BTK (0.67) TDP1BTK
SCHEMBL1322762 0.73 BTK (0.66) BTK
SCHEMBL3968149 0.72 BTK (0.53) BTKSMN1; SMN2KDM4EMEN1POLB
SCHEMBL14270906 0.70 BTK (0.43) TDP1BTKALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081923-A1 CERTAIN SUBSTITUTED AMIDES, METHOD OF MAKING, AND METHOD OF USE THEREOF CGI Pharmaceuticals, Inc. (US) 2009-07-29 EP disclosed
WO-2008033854-A1 CERTAIN SUBSTITUTED AMIDES, METHOD OF MAKING, AND METHOD OF USE THEREOF CGI PHARMACEUTICALS, INC. (US) 2008-03-20 WO disclosed