SCHEMBL3969273

SCHEMBL3969273

Cc1c(NC(=O)c2cc3c(s2)CCCCC3)cccc1-c1c[nH]c(=O)c(N(C)c2ccc(C(=O)O)cn2)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BTK Q06187 18/20 0.46
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
CD69 Q07108 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3956979 0.99 BTK (0.47) BTKALDH1A1HPGDSMN1; SMN2MEN1
SCHEMBL3964067 0.91 BTK (0.44) BTKALDH1A1HPGDSMN1; SMN2MEN1
SCHEMBL3964057 0.88 TDP1 (0.47) BTKALDH1A1HPGDSMN1; SMN2MEN1
SCHEMBL3968149 0.82 BTK (0.53) BTKSMN1; SMN2MEN1POLBRAB9A
SCHEMBL13893940 0.79 BTK (0.53) BTKALDH1A1HPGDSMN1; SMN2MEN1
SCHEMBL1322787 0.75 BTK (0.76) BTKCD69
SCHEMBL1321960 0.74 BTK (0.58) BTKALDH1A1RAB9AKDM4E
SCHEMBL1321911 0.74 BTK (0.77) BTKCD69
SCHEMBL3965260 0.72 BTK (0.46) BTK
SCHEMBL1321976 0.72 BTK (0.57) BTKCD69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081923-A1 CERTAIN SUBSTITUTED AMIDES, METHOD OF MAKING, AND METHOD OF USE THEREOF CGI Pharmaceuticals, Inc. (US) 2009-07-29 EP disclosed
WO-2008033854-A1 CERTAIN SUBSTITUTED AMIDES, METHOD OF MAKING, AND METHOD OF USE THEREOF CGI PHARMACEUTICALS, INC. (US) 2008-03-20 WO disclosed