Bromide

Bromide

SCHEMBL3964464

Br.O=C(O)C1CCCN(C(=O)O)C1

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
TSHR P16473 1/20 0.43
HPGD P15428 1/20 0.43
CA12 O43570 3/20 0.43
CA1 P00915 3/20 0.43
CA2 P00918 3/20 0.43
CA9 Q16790 3/20 0.43
GRM3 Q14832 1/20 0.43
MAPK1 P28482 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAPT P10636 1/20 0.40
HSD11B1 P28845 1/20 0.39
CREBBP Q92793 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2878783 0.98 ALDH1A1 (0.49) ALDH1A1TSHRHPGDCA12CA1
SCHEMBL2880648 0.98 ALDH1A1 (0.49) ALDH1A1TSHRHPGDCA12CA1
SCHEMBL316646 0.98 ALDH1A1 (0.49) ALDH1A1TSHRHPGDCA12CA1
SCHEMBL7357706 0.92 ALDH1A1 (0.48) ALDH1A1TSHRHPGDCA12CA1
SCHEMBL2875175 0.85 NOTUM (0.46) ALDH1A1MAPT
SCHEMBL2875954 0.85 NOTUM (0.46) ALDH1A1MAPT
SCHEMBL652433 0.85 NOTUM (0.46) ALDH1A1MAPT
SCHEMBL25363482 0.82 ALDH1A1 (0.57) ALDH1A1TSHRCA12CA1CA2
SCHEMBL6831699 0.82 ALDH1A1 (0.51) ALDH1A1TSHRHPGDCA12CA1
SCHEMBL3179327 0.82 ALDH1A1 (0.46) ALDH1A1TSHRHPGDCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009033689-A1 PIPERIDONE DERIVATIVES AND MEDICAL USES THEREOF HEINRICH-PETTE-INSTITUT (DE) 2009-03-19 WO disclosed