SCHEMBL3968486

SCHEMBL3968486

COC(=O)c1ccc2c(c1)CCN(Cc1ccccc1)C2

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.69
POLB P06746 1/20 0.58
HPGD P15428 2/20 0.57
CHRM2 P08172 1/20 0.57
HTR1A P08908 1/20 0.57
CHRM3 P20309 1/20 0.57
DRD4 P21917 1/20 0.57
ADRA1D P25100 1/20 0.57
HTR2C P28335 1/20 0.57
ADRA1A P35348 1/20 0.57
ADRA1B P35368 1/20 0.57
DRD3 P35462 1/20 0.57
HTR2B P41595 1/20 0.57
SLC6A3 Q01959 1/20 0.57
TMEM97 Q5BJF2 1/20 0.57
SIGMAR1 Q99720 1/20 0.57
ACHE P22303 1/20 0.56
KDM4E B2RXH2 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
LMNA P02545 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1205833 0.90 ACACB (0.55) ACACBPOLBHPGDHTR1ADRD4
Hydrochloric Acid SCHEMBL3095011 0.89 ACACB (0.54) ACACBPOLBHPGDHTR1ADRD4
SCHEMBL9950571 0.88 ACACB (0.69) ACACBPOLBHPGDDRD3ACHE
SCHEMBL4239488 0.86 MEN1 (0.61) POLBHPGDCHRM2HTR1ACHRM3
SCHEMBL4517559 0.85 ACACB (0.66) ACACBPOLBHPGDACHEKDM4E
Benzylamine SCHEMBL8532295 0.84 LOXL2 (0.56) ACACBHTR1ADRD4HTR2CHTR2B
SCHEMBL1264338 0.84 HDAC6 (0.65) POLBHPGDKDM4ESMN1; SMN2MEN1
SCHEMBL20672151 0.83 TNF (0.64) ACACBPOLBHPGDACHEKDM4E
SCHEMBL1036356 0.83 ACACB (0.63) ACACBPOLBHPGDACHEKDM4E
SCHEMBL20178679 0.83 ACACB (0.59) ACACBCHRM2CHRM3KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009047240-A1 INDOLE DERIVATIVES USEFUL AS PPAR ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO disclosed
WO-2009047240-A1 INDOLE DERIVATIVES USEFUL AS PPAR ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO disclosed