SCHEMBL3971053

SCHEMBL3971053

CCN1CCN(CCCNc2ncc(C)c(-c3cc4ccccc4s3)n2)CC1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 3/20 0.43
HRH3 Q9Y5N1 1/20 0.39
FGFR1 P11362 4/20 0.38
SRC P12931 3/20 0.38
DRD2 P14416 2/20 0.38
EGFR P00533 1/20 0.38
FGFR2 P21802 1/20 0.38
FGFR4 P22455 1/20 0.38
FGFR3 P22607 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
MERTK Q12866 1/20 0.37
HTR2A P28223 1/20 0.36
HTR7 P34969 1/20 0.36
HTR6 P50406 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3965330 0.94 SLC2A1 (0.43) SLC2A1HRH3FGFR1SRCDRD2
SCHEMBL3963837 0.93 FGFR1 (0.44) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL3971739 0.90 VCP (0.46) SLC2A1HRH3FGFR1SRCDRD2
SCHEMBL3965524 0.90 SLC2A1 (0.42) SLC2A1FGFR1SRCDRD2EGFR
SCHEMBL3969374 0.90 LCK (0.41) HRH3FGFR1SRCDRD2EGFR
SCHEMBL3962142 0.84 ACKR3 (0.55) FGFR1DRD2DRD4DRD3
Hydrochloric Acid SCHEMBL3964380 0.83 TACR2 (0.38) HRH3FGFR1SRCDRD2MERTK
SCHEMBL3966578 0.83 FGFR1 (0.50) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL3964127 0.83 FGFR1 (0.44) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL3970084 0.81 FGFR1 (0.45) FGFR1SRCEGFRFGFR2FGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1989200-B1 [4-(BENZO[B]THIOPHEN-2-YL)-PYRIMIDIN-2-YL]-AMINE DERIVATIVES AS IKK-BETA INHIBITORS FOR THE TREATMENT OF CANCER AND INFLAMMATORY DISEASES LILLY CO ELI (US) 2009-07-29 EP disclosed