SCHEMBL3972071

SCHEMBL3972071

CCCCC(N)c1nc(-c2ccc(Br)cc2)nc2ccc(Cl)cc12

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 7/20 0.51
MAPK1 P28482 2/20 0.48
NPC1 O15118 1/20 0.48
HTT P42858 1/20 0.48
RAB9A P51151 1/20 0.48
HSP90AB1 P08238 1/20 0.37
CYP1A1 P04798 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP1B1 Q16678 1/20 0.36
ATM Q13315 1/20 0.36
KDM4E B2RXH2 1/20 0.36
AKR1B10 O60218 1/20 0.35
SLC2A1 P11166 1/20 0.35
ACP1 P24666 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3978931 0.88 KCNH2 (0.42) ADORA3MAPK1NPC1HTTRAB9A
SCHEMBL3972104 0.81 SLC2A1 (0.47) MAPK1HTTKDM4ESLC2A1
SCHEMBL3974309 0.81 NPC1 (0.55) ADORA3MAPK1NPC1HTTRAB9A
SCHEMBL3974635 0.76 ACP1 (0.58) ADORA3MAPK1SLC2A1ACP1
SCHEMBL3977120 0.74 NPC1 (0.49) ADORA3MAPK1NPC1HTTRAB9A
SCHEMBL3972075 0.74 ADORA3 (0.52) ADORA3MAPK1NPC1HTTRAB9A
SCHEMBL3972857 0.72 NPC1 (0.50) ADORA3MAPK1NPC1HTTRAB9A
SCHEMBL3972319 0.70 NPC1 (0.47) ADORA3MAPK1NPC1HTTRAB9A
SCHEMBL27599043 0.70 NPC1 (0.45) ADORA3MAPK1NPC1HTTRAB9A
SCHEMBL3974636 0.70 ADORA3 (0.47) ADORA3MAPK1NPC1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547702-B2 4-amino-quinazolines ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2009-06-16 US disclosed
US-20060019974-A1 Glycoprotein antagonist; anticholesterol agents; cardiovascular disorders; strokes; antiischemic agents ORTHO-MCNEIL PHARMACEUTICALS, INC. 2006-01-26 US disclosed
WO-2004030672-A1 USE OF 4 AMINO-QUINAZOLINES AS ANTI CANCER AGENTS MERCK PATENT GMBH (DE) 2004-04-15 WO disclosed
EP-1318984-A1 4-AMINO-QUINAZOLINES MERCK PATENT GmbH (DE) 2003-06-18 EP disclosed
WO-2002024667-A1 4-AMINO-QUINAZOLINES MERCK PATENT GMBH (DE) 2002-03-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060019974-A1 Glycoprotein antagonist; anticholesterol agents; cardiovascular disorders; strokes; antiischemic agents SERPINA3, APOL1, MGAT3 ADORA3 448/4885MAPK1 3502/4885NPC1 151/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.