SCHEMBL3972559

SCHEMBL3972559

O=C(O)N1CCN(CCOc2ccc(F)cc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 6/20 0.64
LTA4H P09960 2/20 0.60
DRD3 P35462 7/20 0.58
DRD2 P14416 4/20 0.58
HRH1 P35367 2/20 0.56
HRH2 P25021 1/20 0.56
USP2 O75604 1/20 0.55
ALDH1A1 P00352 1/20 0.55
HPGD P15428 1/20 0.55
LMNA P02545 1/20 0.54
HTR1A P08908 1/20 0.53
HTR2A P28223 1/20 0.53
TMEM97 Q5BJF2 1/20 0.53
SIGMAR1 Q99720 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1730306 0.86 LTA4H (0.77) KCNA5LTA4HDRD3DRD2HRH1
SCHEMBL5480208 0.85 KCNA5 (0.74) KCNA5LTA4HDRD3DRD2HRH1
SCHEMBL23301248 0.85 KCNA5 (0.58) KCNA5LTA4HDRD3DRD2ALDH1A1
SCHEMBL19462784 0.85 DRD3 (0.79) KCNA5DRD3DRD2
SCHEMBL6034033 0.85 KCNA5 (0.64) KCNA5LTA4HDRD3DRD2HRH1
SCHEMBL11336991 0.83 HRH2 (0.78) HRH1HRH2ALDH1A1
SCHEMBL11336995 0.83 HRH2 (0.78) HRH1HRH2ALDH1A1
SCHEMBL2236459 0.82 HRH3 (0.57)
SCHEMBL1730771 0.81 HRH2 (0.58) KCNA5LTA4HDRD3DRD2HRH1
SCHEMBL3871235 0.81 CACNA2D1 (0.60) KCNA5LTA4HDRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1988902-A4 PIPERAZINE DERIVATIVES MS SCIENCE CORP (JP) 2009-05-06 EP disclosed
EP-1988902-A2 PIPERAZINE DERIVATIVES M's Science Corporation (JP) 2008-11-12 EP disclosed
WO-2007097871-A2 PIPERAZINE DERIVATIVES M'S SCIENCE CORPORATION (JP) 2007-08-30 WO disclosed