SCHEMBL3973968

SCHEMBL3973968

Cc1cc(-c2nc(Nc3cccc(CN4CCOCC4)c3)nc3[nH]ccc23)sc1CO

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.43
CDK1 P06493 1/20 0.43
JAK3 P52333 6/20 0.41
JAK2 O60674 5/20 0.41
PTK2 Q05397 4/20 0.41
NUAK1 O60285 2/20 0.40
BMPR1B O00238 1/20 0.40
ACVR1 Q04771 1/20 0.40
SIK2 Q9H0K1 1/20 0.40
AURKA O14965 3/20 0.40
CDK2 P24941 2/20 0.40
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
PLK4 O00444 1/20 0.40
JAK1 P23458 1/20 0.40
CSF1R P07333 4/20 0.40
TBK1 Q9UHD2 4/20 0.40
CHEK1 O14757 2/20 0.40
MAP4K4 O95819 2/20 0.40
PAK4 O96013 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13883515 0.91 TTK (0.45) KDRJAK3JAK2PTK2AURKA
SCHEMBL13883581 0.86 KDR (0.41) KDRCDK1JAK3JAK2PTK2
SCHEMBL3974734 0.84 KDR (0.46) KDRCDK1JAK3JAK2PTK2
SCHEMBL3973909 0.77 TTK (0.58) JAK3JAK2PTK2JAK1LRRK2
SCHEMBL3975392 0.76 PDPK1 (0.43) KDRCDK1JAK3JAK2JAK1
SCHEMBL13883504 0.75 TTK (0.45) KDRJAK3JAK2PTK2AURKA
SCHEMBL3970857 0.75 TTK (0.45) KDRJAK3JAK2PTK2AURKA
SCHEMBL3971647 0.74 PDPK1 (0.47) KDRJAK3JAK2PTK2AURKA
Hydrochloric Acid SCHEMBL3974362 0.74 TTK (0.44) KDRJAK3JAK2PTK2AURKA
SCHEMBL4073485 0.74 TTK (0.47) KDRJAK3JAK2PTK2AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009049028-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USE AS JANUS KINASE MODULATORS TARGEGEN INC. (US) 2009-04-16 WO disclosed
WO-2009049028-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USE AS JANUS KINASE MODULATORS TARGEGEN INC. (US) 2009-04-16 WO disclosed