SCHEMBL3977175

SCHEMBL3977175

CS(=O)(=O)N[C@@H](CCCCN)C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
FOLH1 Q04609 1/20 0.39
CA1 P00915 4/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
HPGDS O60760 1/20 0.37
GSR P00390 1/20 0.37
SIRT6 Q8N6T7 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
CPB2 Q96IY4 3/20 0.36
RNPEP Q9H4A4 1/20 0.36
CA2 P00918 3/20 0.36
NPPA P01160 1/20 0.36
MME P08473 1/20 0.36
ACE P12821 1/20 0.36
ECE1 P42892 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8012073 0.86 MMP2 (0.55) ITGB3ITGA2BMMP2MMP9FOLH1
SCHEMBL7331090 0.86 MMP2 (0.55) ITGB3ITGA2BMMP2MMP9FOLH1
SCHEMBL7299119 0.83 FOLH1 (0.37) ITGB3ITGA2BMMP2MMP9FOLH1
SCHEMBL9346130 0.81 ITGB3 (0.40) ITGB3ITGA2BMMP2MMP9FOLH1
SCHEMBL27750390 0.80 MMP2 (0.50) ITGB3ITGA2BMMP2MMP9FOLH1
SCHEMBL21389077 0.79 CA1 (0.35) ITGB3ITGA2BCA1CA12CA9
SCHEMBL21389092 0.79 CA1 (0.35) ITGB3ITGA2BCA1CA12CA9
SCHEMBL1262904 0.77 FOLH1 (0.43) MMP2MMP9FOLH1HPGDSGSR
SCHEMBL13416824 0.77 FOLH1 (0.43) MMP2MMP9FOLH1HPGDSGSR
SCHEMBL7247656 0.75 CA12 (0.42) CA1CA12CA9RNPEPCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2056817-A1 BENZOFURAN AND BENZOTHIOPHENE DERIVATIVES USEFUL IN THE TREATMENT OF CANCERS OF THE CENTRAL NERVOUS SYSTEM Bayer HealthCare AG (DE) 2009-05-13 EP claimed
WO-2008025509-A1 BENZOFURAN AND BENZOTHIOPHENE DERIVATIVES USEFUL IN THE TREATMENT OF CANCERS OF THE CENTRAL NERVOUS SYSTEM BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-03-06 WO claimed