SCHEMBL3980488

SCHEMBL3980488

CCOP(=O)(OCC)C1CN(S(=O)(=O)c2ccc(Nc3nccc(Nc4ccc(F)c(F)c4)n3)cc2)CCC1C(N)CC

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 8/20 0.43
CHUK O15111 7/20 0.43
CDK4 P11802 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
MAPT P10636 3/20 0.37
LMNA P02545 1/20 0.37
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
KDR P35968 1/20 0.36
JAK2 O60674 2/20 0.35
JAK3 P52333 2/20 0.35
SYK P43405 1/20 0.35
TP53 P04637 2/20 0.34
WEE1 P30291 1/20 0.33
ALK Q9UM73 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3300483 0.86 IKBKB (0.43) IKBKBCHUKCDK4CCNE1CDK2
SCHEMBL13392087 0.79 IKBKB (0.46) IKBKBCHUKCDK4CCNE1CDK2
SCHEMBL3302160 0.79 IKBKB (0.47) IKBKBCHUKCDK4CCNE1CDK2
SCHEMBL3302168 0.74 IKBKB (0.44) IKBKBCHUKCDK4CCNE1CDK2
SCHEMBL3303279 0.74 IKBKB (0.51) IKBKBCHUKCDK4CCNE1CDK2
SCHEMBL14020191 0.72 CDK4 (0.40) IKBKBCHUKCDK4CCNE1CDK2
SCHEMBL3306513 0.72 IKBKB (0.51) IKBKBCHUKCDK4CCNE1CDK2
SCHEMBL3299203 0.72 IKBKB (0.51) IKBKBCHUKCDK4CCNE1CDK2
SCHEMBL4440432 0.72 IKBKB (0.38) IKBKBCHUKCDK4CCNE1CDK2
SCHEMBL14020183 0.71 HTR7 (0.43) IKBKBCHUKCDK4CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009056693-A1 NOVEL DERIVATIVES OF N, N'- 2, 4-DIANILINOPYRIMIDINES, PREPARATION THEREOF AS MEDICAMENTS PHARMACEUTICAL COMPOSITIONS AND IN PARTICULAR AS IKK INHIBITORS SANOFI-AVENTIS (FR) 2009-05-07 WO disclosed