SCHEMBL4440432

SCHEMBL4440432

CCCN(C1CCNCC1P(=O)(OCC)OCC)S(=O)(=O)c1ccc(Nc2nccc(Nc3ccc(F)c(F)c3)n2)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
CDK2 P24941 7/20 0.37
CDK4 P11802 5/20 0.37
CCNE1 P24864 1/20 0.37
KDR P35968 2/20 0.35
SYK P43405 1/20 0.35
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
KCNH2 Q12809 1/20 0.34
PRKCI P41743 1/20 0.34
IGF1R P08069 2/20 0.33
FAM20C Q8IXL6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4441619 0.82 IKBKB (0.42) IKBKBCHUKCDK2CDK4CCNE1
SCHEMBL14020182 0.77 IKBKB (0.47) IKBKBCHUKCDK2CDK4CCNE1
SCHEMBL3979898 0.75 MEN1 (0.42) CDK2CDK4CCNE1KDRSYK
SCHEMBL4622742 0.74 IKBKB (0.49) IKBKBCHUKCDK2CDK4CCNE1
SCHEMBL14020190 0.74 CDK2 (0.38) IKBKBCHUKCDK2CDK4CCNE1
Hydrochloric Acid SCHEMBL4880086 0.73 IKBKB (0.49) IKBKBCHUKCDK2CDK4CCNE1
SCHEMBL3300483 0.73 IKBKB (0.43) IKBKBCHUKCDK2CDK4CCNE1
SCHEMBL14020201 0.73 CDK2 (0.38) IKBKBCHUKCDK2CDK4CCNE1
SCHEMBL4623096 0.72 CDK2 (0.47) IKBKBCHUKCDK2CDK4CCNE1
SCHEMBL3980488 0.72 IKBKB (0.43) IKBKBCHUKCDK2CDK4CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118092-A1 NEW N, N'- 2,4-DIANILINOPYRIMIDINE DERIVATIVES, PREPARATION THEREOF AS DRUGS, PHARMACEUTICAL COMPOSITIONS ESSENTIALLY AS IKK INHIBITORS Sanofi-Aventis (FR) 2009-11-18 EP disclosed
WO-2008099073-A1 N, N' -2, 4-DIANILINOPYRIMIDINES PREPARATION AND USE THEREOF AS IKK INHIBITORS PREPARATION AND TEH PHARMACUETICAL COMPOSITIONS THEREOF SANOFI-AVENTIS (FR) 2008-08-21 WO disclosed