SCHEMBL3980924

SCHEMBL3980924

CC(=O)N1CC(C)N(c2nc3c(C(=O)O)cccc3o2)C(C)C1.[LiH]

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 19/20 0.51
KCNH2 Q12809 4/20 0.47
CYP2C19 P33261 1/20 0.47
IDO1 P14902 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1006765 1.00 HTR3A (0.51) HTR3AKCNH2CYP2C19IDO1MAOA
Lithium Ion SCHEMBL1006763 0.89 HTR3A (0.51) HTR3AKCNH2CYP2C19
SCHEMBL1006502 0.87 HTR3A (0.49) HTR3AKCNH2CYP2C19IDO1MAOA
SCHEMBL3984963 0.87 HTR3A (0.52) HTR3AKCNH2CYP2C19
SCHEMBL1005918 0.87 HTR3A (0.52) HTR3AKCNH2CYP2C19
SCHEMBL1005222 0.86 HTR3A (0.47) HTR3AKCNH2CYP2C19
SCHEMBL3981326 0.86 HTR3A (0.47) HTR3AKCNH2CYP2C19
SCHEMBL3990446 0.86 HTR3A (0.51) HTR3AKCNH2CYP2C19
SCHEMBL1005990 0.86 HTR3A (0.51) HTR3AKCNH2CYP2C19
SCHEMBL1006674 0.85 HTR3A (0.49) HTR3AKCNH2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed