SCHEMBL398275

SCHEMBL398275

C=CC1CCN(CC(=O)O)C1=O

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACE P12821 12/20 0.54
FKBP1A P62942 1/20 0.36
POLB P06746 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
MME P08473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL887073 0.85 ACE (0.40) ACE
SCHEMBL16527291 0.85 TSHR (0.42) ACEFKBP1ACYP2C19
SCHEMBL4658185 0.83 ACE (0.37) ACEPOLBKMT2ASMN1; SMN2L3MBTL1
SCHEMBL15320610 0.81 ACE (0.36) ACE
SCHEMBL9485556 0.80 PIK3CD (0.34) ACEKMT2A
SCHEMBL9000514 0.78 CYP3A4 (0.37) KMT2AL3MBTL1
SCHEMBL7355166 0.77 SMN1; SMN2 (0.32) ACEKMT2ASMN1; SMN2LMNA
SCHEMBL8368471 0.77 CHRNA7 (0.35) L3MBTL1
Water SCHEMBL28388741 0.76 ALDH1A1 (0.33) KMT2ASMN1; SMN2LMNA
SCHEMBL9286164 0.76 ACE (0.50) ACEFKBP1APOLBCYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 228 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4719357-A1 COMPOSITIONS COMPRISING SOTORASIB Amgen Inc. (US) 2026-04-08 EP claimed
WO-2024249660-A1 COMPOSITIONS COMPRISING SOTORASIB AMGEN INC. (US) 2024-12-05 WO claimed
EP-2680823-B1 BINDER POWDERS NANO4M LTD (GB) 2024-05-15 EP claimed
EP-4048247-B1 TRANSDERMAL THERAPEUTIC SYSTEM FOR THE TRANSDERMAL ADMINISTRATION OF FINGOLIMOD LTS LOHMANN THERAPIE SYSTEME AG (DE) 2024-04-03 EP claimed
EP-4076382-B1 TRANSDERMAL THERAPEUTIC SYSTEM CONTAINING AGOMELATINE LTS LOHMANN THERAPIE SYSTEME AG (DE) 2024-03-20 EP claimed
EP-3846783-B1 NANOPARTICLES COMPRISING TACROLIMUS LEON NANODRUGS GMBH (DE) 2023-10-18 EP claimed
EP-3826627-B1 ORALLY ADMINISTERABLE PHARMACEUTICAL DOSAGE FORM WITH MODIFIED RELEASE BAYER AG (DE) 2023-10-18 EP claimed
EP-3958344-B1 BINDER RESIN COMPOSITION AND SEPARATOR FOR ELECTROCHEMICAL DEVICE COMPRISING THE SAME LG ENERGY SOLUTION LTD (KR) 2023-09-27 EP claimed
EP-3996688-B1 PHARMACEUTICAL PREPARATION MERCK PATENT GMBH (DE) 2023-09-06 EP claimed
EP-3281626-B1 SOLUBLE MICRONEEDLE FOR DELIVERING POORLY-SOLUBLE DRUG LG HOUSEHOLD & HEALTH CARE LTD (KR) 2023-08-23 EP claimed
EP-0289977-B1 SUSTAINED-RELEASE ORAL ADMINISTRATION FORMS CIBA-GEIGY AG (CH) 1993-09-15 EP claimed
EP-0557489-A1 COMPOSITION PROVIDING A LASTING COSMETIC AND/OR PHARMACEUTICAL TREATMENT OF THE UPPER EPIDERMAL LAYERS BY TOPICAL APPLICATION ON THE SKIN. OREAL (FR) 1993-09-01 EP claimed
WO-1993005753-A1 COMPOSITION PROVIDING A LASTING COSMETIC AND/OR PHARMACEUTICAL TREATMENT OF THE UPPER EPIDERMAL LAYERS BY TOPICAL APPLICATION ON THE SKIN L'OREAL (FR) 1993-04-01 WO claimed
EP-0248062-B1 MEDICAMENTS Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 1992-05-06 EP claimed
EP-0277092-B1 THERAPEUTIC SYSTEM FOR SLIGHTLY SOLUBLE ACTIVE INGREDIENTS CIBA-GEIGY AG (CH) 1992-01-29 EP claimed
EP-0165397-B1 HAIR CARE COMPOSITIONS Revlon, Inc. (US) 1991-07-17 EP claimed
EP-0248047-B1 MEDICAMENT WITH ANTI-TUMORAL ACTION CONTAINING HEXADECYLPHOSPHOCHOLINE Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 1991-06-19 EP claimed
EP-0164967-B1 PHARMACEUTICAL COMPOSITION OF SPARINGLY SOLUBLE MEDICAMENT AND METHOD FOR ITS PREPARATION STERWIN AG. (CH) 1990-09-12 EP claimed
EP-0213999-B1 COSMETIC COMPOSITION OBTAINED FROM CONNECTIVE TISSUE CELL CULTURES Seguin, Marie-Christine (MC) 1990-01-03 EP claimed
EP-0213999-A1 Cosmetic composition obtained from connective tissue cell cultures Seguin, Marie-Christine (MC) 1987-03-11 EP claimed