SCHEMBL3983192

SCHEMBL3983192

O=C(NNC(=O)c1occ(-c2ccccc2)c1-c1ccccc1)c1ccc(O)c(F)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
GCGR P47871 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
HSD17B10 Q99714 1/20 0.39
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3981613 0.89 CCNC (0.42) MEN1KMT2ANPC1RAB9ACTDSP1
SCHEMBL3982429 0.89 TOP1 (0.44) MEN1KMT2ANPC1RAB9ACTDSP1
SCHEMBL3983962 0.86 MEN1 (0.40) MEN1KMT2ANPC1RAB9ACTDSP1
SCHEMBL3982131 0.86 KMT2A (0.40) ESR2MEN1KMT2ANPC1RAB9A
SCHEMBL3981075 0.86 MEN1 (0.40) MEN1KMT2ANPC1RAB9ACTDSP1
SCHEMBL3973507 0.86 MEN1 (0.40) MEN1KMT2ANPC1RAB9ACTDSP1
SCHEMBL3978766 0.85 PLK1 (0.38) MEN1KMT2ANPC1RAB9ACTDSP1
SCHEMBL3982336 0.84 LMNA (0.47) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL3977724 0.83 NPC1 (0.50) MEN1KMT2ANPC1RAB9ACTDSP1
SCHEMBL3975924 0.83 GRM5 (0.41) MEN1KMT2AGCGRKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7514452-B2 2-furancarboxylic acid hydrazides and pharmaceutical compositions containing the same DAINIPPON PHARMACEUTICAL CO., LTD (JP) 2009-04-07 US disclosed
US-20050171196-A1 2-Furancarboxylic acid hydrazides and pharmaceutical compositions containing the same DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2005-08-04 US disclosed
EP-1489077-A1 2-FURANCARBOXYLIC ACID HYDRAZIDES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 2004-12-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050171196-A1 2-Furancarboxylic acid hydrazides and pharmaceutical compositions containing the same GLP1R, GCGR, GPR119 ESR1 503/4885ESR2 432/4885MEN1 1481/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.