SCHEMBL3983860

SCHEMBL3983860

CCN(Cc1ccc(C#CCCO)cc1)c1cccc2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.38
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
LMNA P02545 2/20 0.37
HTT P42858 2/20 0.37
HPGD P15428 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
HRH3 Q9Y5N1 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 5/20 0.36
MEN1 O00255 4/20 0.36
ACACB O00763 1/20 0.35
MAPT P10636 1/20 0.35
POLB P06746 1/20 0.35
CNR2 P34972 1/20 0.34
NPC1 O15118 1/20 0.34
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB1 P18505 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3988560 0.90 SIGMAR1 (0.39) SIGMAR1ALDH1A1KDM4ELMNAHTT
SCHEMBL3987757 0.82 TSHR (0.57) ALDH1A1KDM4ELMNAHPGDL3MBTL1
SCHEMBL3992396 0.79 SIGMAR1 (0.41) SIGMAR1ALDH1A1KDM4ELMNAHTT
SCHEMBL9086683 0.78 SIGMAR1 (0.46) SIGMAR1ALDH1A1KDM4ELMNAHTT
SCHEMBL2343211 0.77 TSHR (0.59) SIGMAR1ALDH1A1KDM4ELMNAHTT
SCHEMBL3983733 0.77 KDM4E (0.39) SIGMAR1ALDH1A1KDM4ELMNAHTT
Hydrochloric Acid SCHEMBL3792219 0.76 TSHR (0.58) SIGMAR1ALDH1A1KDM4ELMNAHTT
SCHEMBL3989721 0.73 KDM4E (0.41) SIGMAR1ALDH1A1KDM4ELMNAHTT
SCHEMBL3991413 0.72 ALDH1A1 (0.42) SIGMAR1ALDH1A1KDM4ELMNAHTT
Hydrochloric Acid SCHEMBL7967252 0.72 CNR2 (0.46) SIGMAR1ALDH1A1KDM4ELMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061449-A1 SUBSTITUTED ACETYLENIC COMPOUNDS USEFUL FOR THE TREATMENT OF DISEASES Leo Pharma A/S (DK) 2009-05-27 EP disclosed
WO-2008019690-A1 SUBSTITUTED ACETYLENIC COMPOUNDS USEFUL FOR THE TREATMENT OF DISEASES LEO PHARMA A/S (DK) 2008-02-21 WO disclosed