SCHEMBL3984677

SCHEMBL3984677

COC(=O)c1cccc2oc(N3C(C)CNCC3C)nc12

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 13/20 0.61
KCNH2 Q12809 3/20 0.61
CYP2C19 P33261 1/20 0.61
TOP2A P11388 2/20 0.47
RIPK1 Q13546 1/20 0.39
PKN1 Q16512 1/20 0.37
PKN2 Q16513 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1004565 1.00 HTR3A (0.61) HTR3AKCNH2CYP2C19TOP2ARIPK1
SCHEMBL1005020 0.87 HTR3A (0.62) HTR3AKCNH2CYP2C19TOP2A
Lithium Ion SCHEMBL1006319 0.86 HTR3A (0.61) HTR3AKCNH2CYP2C19
SCHEMBL1006321 0.86 HTR3A (0.61) HTR3AKCNH2CYP2C19TOP2A
SCHEMBL1005918 0.84 HTR3A (0.52) HTR3AKCNH2CYP2C19TOP2A
SCHEMBL3984963 0.84 HTR3A (0.52) HTR3AKCNH2CYP2C19TOP2A
SCHEMBL3990444 0.82 HTR3A (0.49) HTR3AKCNH2CYP2C19TOP2A
SCHEMBL1005434 0.82 HTR3A (0.49) HTR3AKCNH2CYP2C19TOP2A
SCHEMBL1006097 0.81 HTR3A (0.51) HTR3AKCNH2CYP2C19TOP2AKDM4E
SCHEMBL3988561 0.81 HTR3A (0.51) HTR3AKCNH2CYP2C19TOP2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed