SCHEMBL3984732

SCHEMBL3984732

Cc1ccc2oc(N3CCCC3C(N)=O)nc2c1C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ELANE P08246 2/20 0.52
PIK3CA P42336 6/20 0.39
MAT2A P31153 2/20 0.37
RAB9A P51151 2/20 0.36
HSD17B10 Q99714 1/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
PIK3CD O00329 1/20 0.35
PIK3CG P48736 1/20 0.35
AR P10275 1/20 0.34
POLB P06746 1/20 0.34
LMNA P02545 1/20 0.34
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3985869 0.80 ELANE (0.56) ELANEMAT2AHSD17B10
SCHEMBL1005780 0.75 HTR3A (0.49) PIK3CA
SCHEMBL1006741 0.75 HTR3A (0.49) PIK3CA
SCHEMBL1003484 0.74 ELANE (0.50) ELANEHSD17B10
SCHEMBL1003486 0.74 ELANE (0.50) ELANEHSD17B10
SCHEMBL3984179 0.73 HTR3A (0.35) ALDH1A1POLB
SCHEMBL1004322 0.73 HTR3A (0.51) PIK3CARAB9ANPC1
SCHEMBL1005156 0.73 HTR3A (0.51) PIK3CARAB9ANPC1
SCHEMBL1006071 0.72 HTR3A (0.51) ALDH1A1POLB
SCHEMBL1006356 0.72 HTR3A (0.52) ALDH1A1PIK3CDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed