SCHEMBL3985840

SCHEMBL3985840

Cc1[c]nc(-c2cccc(CO)c2)o1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.45
KDR P35968 2/20 0.41
MAP2K4 P45985 2/20 0.41
S1PR1 P21453 1/20 0.41
S1PR3 Q99500 1/20 0.41
ACMSD Q8TDX5 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA7 P36544 1/20 0.39
ATR Q13535 2/20 0.38
NOTUM Q6P988 1/20 0.38
DHODH Q02127 1/20 0.38
HTR1A P08908 1/20 0.36
GPR68 Q15743 1/20 0.36
FLT1 P17948 1/20 0.36
FLT4 P35916 1/20 0.36
CDK8 P49336 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
VSIR Q9H7M9 1/20 0.36
PDE10A Q9Y233 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1435654 0.79 RAB9A (0.54) NOTUM
SCHEMBL1435603 0.76 NPC1 (0.51) NOTUM
SCHEMBL504678 0.75 NPC1 (0.47) NOTUM
SCHEMBL2026858 0.74 MET (0.50) PRKCIKDRMAP2K4S1PR1S1PR3
SCHEMBL19679762 0.74 HPGD (0.66) PRKCIMAP2K4S1PR3ATR
SCHEMBL30018059 0.71 S1PR1 (0.56) PRKCIKDRMAP2K4S1PR1S1PR3
SCHEMBL22469950 0.71 S1PR1 (0.56) PRKCIKDRMAP2K4S1PR1S1PR3
SCHEMBL504247 0.70 CYP1A2 (0.55) S1PR1NOTUM
SCHEMBL4191589 0.70 PRKCI (0.72) PRKCIMAP2K4ACMSDCHRNB4CHRNA3
SCHEMBL11644463 0.70 KDM4E (0.56) KDRVSIRPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7473705-B2 Hexafluoroisopropanol substituted ether derivatives HOFFMANN-LA ROCHE INC. (US) 2009-01-06 US claimed
EP-1802566-B1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-11-26 EP claimed
EP-1802566-A1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-07-04 EP claimed
WO-2006037480-A1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2006-04-13 WO claimed
US-20060074115-A1 Novel hexafluoroisopropanol substituted ether derivatives HOFFMANN-LA ROCHE INC. 2006-04-06 US claimed
US-7473705-B2 Hexafluoroisopropanol substituted ether derivatives HOFFMANN-LA ROCHE INC. (US) 2009-01-06 US disclosed
EP-1802566-B1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-11-26 EP disclosed
US-20060074115-A1 Novel hexafluoroisopropanol substituted ether derivatives HOFFMANN-LA ROCHE INC. 2006-04-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060074115-A1 Novel hexafluoroisopropanol substituted ether derivatives NR1H3, NR1H2, NR1I2 PRKCI 1593/4885KDR 1157/4885MAP2K4 4340/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.