SCHEMBL3986750

SCHEMBL3986750

C[Si](C)(C)C#Cc1ccc(CNCCc2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.57
MAPT P10636 1/20 0.57
BCHE P06276 5/20 0.52
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
OPRM1 P35372 1/20 0.48
ATM Q13315 1/20 0.48
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA4 P22748 1/20 0.48
CA9 Q16790 1/20 0.48
SIGMAR1 Q99720 3/20 0.46
TDP1 Q9NUW8 1/20 0.46
EPHX2 P34913 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
LTA4H P09960 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3986690 0.86 GAA (0.50) GAAMAPTBCHEMEN1KMT2A
SCHEMBL3988576 0.84 GAA (0.69) GAAMAPTBCHEMEN1KMT2A
SCHEMBL3982330 0.80 HPGD (0.47) BCHEMEN1KMT2ACA12CA1
SCHEMBL3272134 0.79 GAA (0.91) GAAMAPTBCHEMEN1KMT2A
SCHEMBL11881258 0.79 GAA (0.91) GAAMAPTBCHEMEN1KMT2A
SCHEMBL30707909 0.78 LOXL2 (0.36) MEN1KMT2AALDH1A1TDP1SMN1; SMN2
SCHEMBL27228 0.77 GAA (0.95) GAAMAPTBCHEMEN1KMT2A
SCHEMBL3982245 0.76 GAA (0.67) GAAMAPTBCHEMEN1KMT2A
SCHEMBL3040879 0.76 S1PR1 (0.54) ALDH1A1
Ammonia Solution, Strong SCHEMBL23581968 0.75 GAA (0.91) GAAMAPTBCHEMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061449-A1 SUBSTITUTED ACETYLENIC COMPOUNDS USEFUL FOR THE TREATMENT OF DISEASES Leo Pharma A/S (DK) 2009-05-27 EP disclosed
WO-2008019690-A1 SUBSTITUTED ACETYLENIC COMPOUNDS USEFUL FOR THE TREATMENT OF DISEASES LEO PHARMA A/S (DK) 2008-02-21 WO disclosed