SCHEMBL3987553

SCHEMBL3987553

CN(Cc1ccc(Cl)cc1)C(=O)[C@H]1CCCN1C(=O)OC(C)(C)C

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 16/20 0.66
ALDH1A1 P00352 1/20 0.53
USP30 Q70CQ3 1/20 0.51
CPT2 P23786 1/20 0.48
CPT1A P50416 1/20 0.48
PKM P14618 1/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3987554 1.00 CCR1 (0.66) CCR1ALDH1A1USP30CPT2CPT1A
SCHEMBL7311067 0.89 CPT2 (0.61) CCR1ALDH1A1USP30CPT2CPT1A
SCHEMBL3984104 0.86 CCR1 (0.67) CCR1ALDH1A1CPT2CPT1APKM
SCHEMBL3984106 0.86 CCR1 (0.67) CCR1ALDH1A1CPT2CPT1APKM
SCHEMBL3981116 0.85 CCR1 (0.57) CCR1ALDH1A1USP30
SCHEMBL3981118 0.85 CCR1 (0.57) CCR1ALDH1A1USP30
SCHEMBL13769199 0.82 ALDH1A1 (0.51) CCR1ALDH1A1USP30
SCHEMBL31630412 0.81 ALDH1A1 (0.47) CCR1ALDH1A1USP30
SCHEMBL13769344 0.81 ALDH1A1 (0.50) CCR1ALDH1A1USP30
SCHEMBL3987624 0.81 CCR1 (0.69) CCR1CPT2CPT1APKMHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2059502-A2 PROLINE UREA CCR1 ANTAGONISTS FOR THE TREATMENT OF AUTOIMMUNE DISEASES OR INFLAMMATION LIGAND PHARMACEUTICALS INCORPORATED (US) 2009-05-20 EP disclosed
WO-2008011392-A2 PROLINE UREA CCR1 ANTAGONISTS FOR THE TREATMENT OF AUTOIMMUNE DISEASES OR INFLAMMATION LIGAND PHARMACUETICALS INCORPORATED (US) 2008-01-24 WO disclosed