SCHEMBL3987624

SCHEMBL3987624

CN(Cc1ccc(Cl)cc1)C(=O)[C@H]1CCCN1C(N)=S

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 17/20 0.69
PKM P14618 1/20 0.51
HTT P42858 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
CPT2 P23786 1/20 0.48
CPT1A P50416 1/20 0.48
TACR1 P25103 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3984104 0.82 CCR1 (0.67) CCR1PKMHTTSMN1; SMN2CPT2
SCHEMBL3984106 0.82 CCR1 (0.67) CCR1PKMHTTSMN1; SMN2CPT2
SCHEMBL9910985 0.81 CCR1 (0.73) CCR1PKMHTTSMN1; SMN2CPT2
SCHEMBL14306232 0.81 CCR1 (0.75) CCR1CPT2CPT1A
SCHEMBL3987554 0.81 CCR1 (0.66) CCR1PKMHTTSMN1; SMN2CPT2
SCHEMBL3987553 0.81 CCR1 (0.66) CCR1PKMHTTSMN1; SMN2CPT2
SCHEMBL14304108 0.81 CCR1 (0.71) CCR1PKMHTTSMN1; SMN2CPT2
SCHEMBL14313691 0.79 CCR1 (0.72) CCR1PKMHTTSMN1; SMN2CPT2
SCHEMBL14306239 0.78 CCR1 (0.92) CCR1
SCHEMBL14304103 0.78 CCR1 (1.00) CCR1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2059502-A2 PROLINE UREA CCR1 ANTAGONISTS FOR THE TREATMENT OF AUTOIMMUNE DISEASES OR INFLAMMATION LIGAND PHARMACEUTICALS INCORPORATED (US) 2009-05-20 EP disclosed
WO-2008011392-A2 PROLINE UREA CCR1 ANTAGONISTS FOR THE TREATMENT OF AUTOIMMUNE DISEASES OR INFLAMMATION LIGAND PHARMACUETICALS INCORPORATED (US) 2008-01-24 WO disclosed