SCHEMBL3987602

SCHEMBL3987602

COc1ccc(COC(c2cc(C)c(OCCO)c(C)c2)(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APP P05067 7/20 0.41
SCN8A Q9UQD0 1/20 0.38
BRD4 O60885 1/20 0.36
PPARD Q03181 1/20 0.35
IDH1 O75874 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
IDO1 P14902 2/20 0.34
AGXT P21549 2/20 0.34
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
HTR7 P34969 1/20 0.34
ADRA1A P35348 1/20 0.34
FFAR4 Q5NUL3 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3982029 0.94 APP (0.40) APPSCN8APPARDIDH1IDO1
SCHEMBL3979075 0.85 APP (0.51) APPNPC1POLBRAB9ASMN1; SMN2
SCHEMBL3987085 0.83 MAPT (0.48) NPC1POLBRAB9ASMN1; SMN2
SCHEMBL3984342 0.82 APP (0.43) APPNPC1RAB9A
SCHEMBL3978166 0.82 ALOX5 (0.43) APPIDH1IDO1AGXT
SCHEMBL5906907 0.81 CA1 (0.36) APPIDH1IDO1AGXT
SCHEMBL3979486 0.81 PPARD (0.42) APPPPARDPTGDR2FFAR4
SCHEMBL3983212 0.78 IGF1R (0.40) IDH1IDO1AGXT
SCHEMBL3983187 0.77 APP (0.42) APPNPC1RAB9A
SCHEMBL3979249 0.75 CALM1 (0.50) APPIDO1AGXTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7473705-B2 Hexafluoroisopropanol substituted ether derivatives HOFFMANN-LA ROCHE INC. (US) 2009-01-06 US disclosed
EP-1802566-B1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-11-26 EP disclosed
EP-1802566-A1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-07-04 EP disclosed
WO-2006037480-A1 HEXAFLUOROISOPROPANOL SUBSTITUTED ETHER DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2006-04-13 WO disclosed
US-20060074115-A1 Novel hexafluoroisopropanol substituted ether derivatives HOFFMANN-LA ROCHE INC. 2006-04-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060074115-A1 Novel hexafluoroisopropanol substituted ether derivatives NR1H3, NR1H2, NR1I2 APP 1609/4885SCN8A 1741/4885BRD4 1181/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.