SCHEMBL3994033

SCHEMBL3994033

CN(Cc1nc2ccccc2n1CCCN1CCN(C(=O)O)CC1)C1CCCc2cccnc21

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 19/20 0.71
CHRM2 P08172 1/20 0.45
CHRM4 P08173 1/20 0.45
CHRM5 P08912 1/20 0.45
CYP2D6 P10635 1/20 0.45
CHRM1 P11229 1/20 0.45
CHRM3 P20309 1/20 0.45
CYP3A4 P08684 1/20 0.45
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4934665 0.91 CXCR4 (0.79) CXCR4KCNH2
SCHEMBL4940872 0.90 CXCR4 (0.66) CXCR4CHRM2CHRM4CHRM5CYP2D6
SCHEMBL4001138 0.88 CXCR4 (0.65) CXCR4
SCHEMBL4936708 0.87 CXCR4 (0.76) CXCR4CYP3A4KCNH2
SCHEMBL4938038 0.87 CXCR4 (0.76) CXCR4CHRM2CHRM4CHRM5CYP2D6
SCHEMBL3993468 0.87 CXCR4 (0.69) CXCR4KCNH2
SCHEMBL4935692 0.84 CXCR4 (0.76) CXCR4KCNH2
SCHEMBL3993485 0.84 CXCR4 (0.73) CXCR4KCNH2
SCHEMBL3996935 0.84 CXCR4 (0.69) CXCR4KCNH2
SCHEMBL3990885 0.84 CXCR4 (0.70) CXCR4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778231-A4 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2009-06-03 EP disclosed
EP-1778231-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-02 EP disclosed
WO-2006020415-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-02-23 WO disclosed