SCHEMBL4940872

SCHEMBL4940872

CN(Cc1nc2ccccc2n1CCCN1CCN(C(=O)OC(C)(C)C)CC1)C1CCCc2cccnc21

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 19/20 0.66
CHRM2 P08172 1/20 0.44
CHRM4 P08173 1/20 0.44
CHRM5 P08912 1/20 0.44
CYP2D6 P10635 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3994033 0.90 CXCR4 (0.71) CXCR4CHRM2CHRM4CHRM5CYP2D6
SCHEMBL4276762 0.89 CXCR4 (0.60) CXCR4
SCHEMBL4940055 0.88 CXCR4 (0.64) CXCR4
SCHEMBL4934665 0.87 CXCR4 (0.79) CXCR4
SCHEMBL4939479 0.87 CXCR4 (0.63) CXCR4
SCHEMBL4935750 0.85 CXCR4 (0.65) CXCR4
SCHEMBL3998366 0.85 CXCR4 (0.66) CXCR4
SCHEMBL4939959 0.85 CXCR4 (0.74) CXCR4
SCHEMBL4935802 0.84 CXCR4 (0.70) CXCR4
SCHEMBL4933459 0.84 CXCR4 (0.61) CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080096861-A1 Chemical Compounds SMITHKLINE BEECHAM CORPORATION (US) 2008-04-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080096861-A1 Chemical Compounds CCR5, CXCR4, CXCR3 CXCR4 2/4885CHRM2 3578/4885CHRM4 1640/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.