SCHEMBL3997883

SCHEMBL3997883

C=CCOc1ccc(CN2CCC(N(c3cnc4ccccc4c3)N(c3cnc4ccccc4c3)C3CCN(Cc4ccc(OC(C)C)c(OCC)c4)CC3)CC2)cc1OCC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 16/20 0.43
HRH1 P35367 3/20 0.43
HTR2B P41595 2/20 0.43
DRD2 P14416 2/20 0.39
DRD4 P21917 2/20 0.39
DRD3 P35462 2/20 0.39
GMNN O75496 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
HPGD P15428 1/20 0.39
PMP22 Q01453 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
POLB P06746 1/20 0.38
DRD1 P21728 1/20 0.37
HTR2A P28223 1/20 0.37
SIGMAR1 Q99720 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3996567 0.90 SSTR5 (0.46) SSTR5HRH1HTR2BDRD2DRD4
SCHEMBL4000428 0.84 SSTR5 (0.56) SSTR5HRH1HTR2BALDH1A1ABCB1
SCHEMBL3993879 0.84 SSTR5 (0.45) SSTR5HRH1HTR2BALDH1A1ABCB1
SCHEMBL4002555 0.82 NPC1 (0.43) SSTR5HRH1HTR2BALDH1A1LMNA
SCHEMBL4002561 0.81 DRD2 (0.45) SSTR5HRH1HTR2BDRD2CYP3A4
SCHEMBL1878273 0.81 SSTR5 (0.56) SSTR5HRH1HTR2B
SCHEMBL1878673 0.81 SSTR5 (0.56) SSTR5HRH1HTR2B
SCHEMBL4002203 0.80 SSTR5 (0.53) SSTR5HRH1HTR2BDRD2DRD4
SCHEMBL4002214 0.79 SSTR5 (0.50) SSTR5HRH1HTR2BALDH1A1ABCB1
SCHEMBL3999810 0.79 SSTR5 (0.49) SSTR5HRH1HTR2BDRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2066658-A1 PYRIDINE- AND QUINOLINE-PYRIMIDINE-DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2009-06-10 EP claimed
WO-2008031735-A1 PYRIDINE- AND QUINOLINE-PYRIMIDINE-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-03-20 WO claimed