SCHEMBL4000428

SCHEMBL4000428

CCOc1cc(CN2CCC(N(c3cnc4ccccc4c3)N(c3cnc4ccccc4c3)C3CCN(Cc4ccc(OCC)c(OCC)c4)CC3)CC2)ccc1OC

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 12/20 0.56
HRH1 P35367 1/20 0.56
HTR2B P41595 1/20 0.56
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
ABCB1 P08183 1/20 0.47
KCNH2 Q12809 1/20 0.47
BCHE P06276 1/20 0.46
ACHE P22303 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4002214 0.89 SSTR5 (0.50) SSTR5HRH1HTR2BKMT2AKDM4E
SCHEMBL3996567 0.86 SSTR5 (0.46) SSTR5HRH1HTR2BALDH1A1ABCB1
SCHEMBL4002555 0.85 NPC1 (0.43) SSTR5HRH1HTR2BKMT2AKDM4E
SCHEMBL3993879 0.85 SSTR5 (0.45) SSTR5HRH1HTR2BKMT2AKDM4E
SCHEMBL3996819 0.85 SSTR5 (0.48) SSTR5HRH1HTR2BKMT2AMEN1
SCHEMBL3997883 0.84 SSTR5 (0.43) SSTR5HRH1HTR2BALDH1A1ABCB1
SCHEMBL4002203 0.84 SSTR5 (0.53) SSTR5HRH1HTR2BKMT2AALDH1A1
SCHEMBL3997486 0.83 SSTR5 (0.52) SSTR5HRH1HTR2BKCNH2
SCHEMBL4002561 0.83 DRD2 (0.45) SSTR5HRH1HTR2BKMT2AMEN1
SCHEMBL4000512 0.81 SSTR5 (0.46) SSTR5HRH1HTR2BKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2066658-A1 PYRIDINE- AND QUINOLINE-PYRIMIDINE-DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2009-06-10 EP claimed
WO-2008031735-A1 PYRIDINE- AND QUINOLINE-PYRIMIDINE-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-03-20 WO claimed