Captopril

Captopril

SCHEMBL4

C[C@H](CS)C(=O)N1CCC[C@H]1C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACE

The experimentally established mechanism targets of Captopril. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACE known ✓ P12821 7/20 1.00
REN P00797 4/20 1.00
KDM4E B2RXH2 1/20 1.00
F2 P00734 1/20 1.00
LMNA P02545 1/20 1.00
LTA4H P09960 1/20 1.00
MAPT P10636 1/20 1.00
PEPD P12955 1/20 1.00
ALOX15 P16050 1/20 1.00
PTGS1 P23219 1/20 1.00
HTR2A P28223 1/20 1.00
PTGS2 P35354 1/20 1.00
HRH1 P35367 1/20 1.00
THPO P40225 1/20 1.00
PMP22 Q01453 1/20 1.00
HSD17B10 Q99714 1/20 1.00
ACE2 Q9BYF1 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
D-Captopril SCHEMBL7983782 1.00 ACE (1.00) ACERENKDM4EF2LMNA
D-Captopril SCHEMBL675797 1.00 ACE (1.00) ACERENKDM4EF2LMNA
D-Captopril SCHEMBL2444049 1.00 ACE (1.00) ACERENKDM4EF2LMNA
D-Captopril SCHEMBL678794 1.00 ACE (1.00) ACERENKDM4EF2LMNA
D-Captopril SCHEMBL1913521 1.00 ACE (1.00) ACERENKDM4EF2LMNA
D-Captopril SCHEMBL2422871 1.00 ACE (1.00) ACERENKDM4EF2LMNA
D-Captopril SCHEMBL2444053 1.00 ACE (1.00) ACERENKDM4EF2LMNA
Captopril SCHEMBL2786691 1.00 ACE (1.00) ACERENKDM4EF2LMNA
Captopril SCHEMBL5556542 0.98 ACE (0.97) ACERENKDM4EF2LMNA
Captopril SCHEMBL2489188 0.98 ACE (0.97) ACERENKDM4EF2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 72891 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4747611-A1 OPTICAL ELECTRODE ANALYTE DETECTION SYSTEM AND METHODS OF USE Vital Biosciences Inc. (CA) 2026-05-27 EP claimed
EP-3607938-B1 PHARMACEUTICAL COMPOSITION SOVIC BRKICIC LJILJANA (HR) 2026-05-27 EP claimed
EP-4743449-A1 L-ARGININE SALT OF 4-CHLORO-5-[4-(2,6-DICHLOROPHENYL)SULFONYLPIPERAZIN-1-YL]-1-BENZOFURAN-2-CARBOXYLIC ACID AND VARIOUS FORMS THEREOF ENYO Pharma (FR) 2026-05-20 EP claimed
EP-4743450-A1 L-LYSINE SALT OF 4-CHLORO-5-[4-(2,6-DICHLOROPHENYL)SULFONYLPIPERAZIN-1-YL]-1-BENZOFURAN-2-CARBOXYLIC ACID AND VARIOUS FORMS THEREOF ENYO Pharma (FR) 2026-05-20 EP claimed
EP-4743451-A1 TROMETHAMINE SALT OF 4-CHLORO-5-[4-(2,6-DICHLOROPHENYL)SULFONYLPIPERAZIN-1-YL]-1-BENZOFURAN-2-CARBOXYLIC ACID AND VARIOUS FORMS THEREOF ENYO Pharma (FR) 2026-05-20 EP claimed
CN-122059859-A Synthesis method of diaryl methyl sulfide under biocompatible condition 南京工业大学 2026-05-19 CN claimed
EP-4739293-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF AUTOIMMUNE DISORDERS AZURA OPHTHALMICS LTD (IL) 2026-05-13 EP claimed
EP-4739291-A2 ADMINISTRATION OF KERATOLYTICS TO OCULAR AND PERIOCULAR SURFACES AZURA OPHTHALMICS LTD (IL) 2026-05-13 EP claimed
CN-122010656-A Application of oxyalkylisourea in introducing methyl and isotopically-labeled methyl 陕西师范大学 2026-05-12 CN claimed
US-20260124148-A1 POLYPEPTIDE FORMULATIONS FOR ORAL DELIVERY BHAMIS RES LABORATORY PVT LTD (IN) 2026-05-07 US claimed
EP-0072868-A1 CYCLODEXTRIN CLATHRATE COMPOUNDS OF SULFUR-CONTAINING COMPOUNDS SANTEN PHARMACEUTICAL CO., LTD. (JP) 1983-03-02 EP claimed
US-4369172-A Prolonged release therapeutic compositions based on hydroxypropylmethylcellulose FOREST LABORATORIES INC. (US) 1983-01-18 US claimed
EP-0055870-A1 Pyridylmethyl esters of selected bio-affecting carboxylic acids, process for preparing and pharmaceutical composition comprising the same MERCK & CO. INC. (US) 1982-07-14 EP claimed
US-4332726-A Purification of mercaptoacyl amino acids E. R. SQUIBB & SONS, INC. (US) 1982-06-01 US claimed
EP-0051278-A1 Soft tertiary amine esters of bio-affecting carboxylic acids, processes for preparing and a pharmaceutical composition containing the same MERCK & CO. INC. (US) 1982-05-12 EP claimed
EP-0048159-A2 Novel carboxyalkyl peptides and thioethers and ethers of peptides as antihypertensive agents UNIVERSITY OF MIAMI (US) 1982-03-24 EP claimed
US-4307099-A Reaction products of pyrazolo[1,5-c]quinazoline derivatives and proline derivatives and methods for reducing blood pressure while inhibiting allergic reactions with them E. R. SQUIBB & SONS, INC. (US) 1981-12-22 US claimed
US-4297282-A REACTING AN A-METHYL-B-ACYLTHIOPROPIONIC ACID WITH AN OPTICALLY ACTIVE ARYLALKYL PRIMARY AMINE; CRYSTALLIZATION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1981-10-27 US claimed
EP-0036145-A1 An orally administered drug form comprising a polar bioactive agent and an adjuvant INTERx RESEARCH CORPORATION (US) 1981-09-23 EP claimed
EP-0031561-A2 A rectally administered suppository comprising a drug and an adjuvant MERCK & CO. INC. (US) 1981-07-08 EP claimed