SCHEMBL4000359

SCHEMBL4000359

B.CCc1cccnc1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.44
FFAR1 O14842 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA1 P14867 2/20 0.39
GABRB2 P47870 2/20 0.39
CYP2C9 P11712 1/20 0.39
NAMPT P43490 1/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HTR1A P08908 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
SLC40A1 Q9NP59 1/20 0.37
CYP1A2 P05177 1/20 0.37
MAPT P10636 1/20 0.37
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
KMT2A Q03164 1/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL487765 0.98
SCHEMBL31421766 0.98
Bromide SCHEMBL28265555 0.95 P2RX7 (0.44) P2RX7FFAR1GABRA5GABRA1GABRB2
Acetic Acid SCHEMBL28688767 0.88 P2RX7 (0.47) P2RX7FFAR1GABRA1GABRB2CYP2C9
Acetic Acid SCHEMBL7435578 0.86 P2RX7 (0.46) P2RX7FFAR1GABRA1GABRB2CYP2C9
SCHEMBL10750692 0.86 NMT1 (0.42) P2RX7FFAR1GABRA5GABRA1GABRB2
SCHEMBL2650778 0.82
SCHEMBL7075262 0.80 GRM5 (0.50) P2RX7FFAR1GABRA5CYP2C9NAMPT
SCHEMBL22931645 0.79 VHL (0.44) P2RX7KDM4EALDH1A1MKNK1MKNK2
SCHEMBL904436 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110520127-A Piperidinyl-substituted and piperazinyl-substituted heteroaromatic carboxamides as modulators of GPR6 TAKEDA PHARMACEUTICALS CO 2019-11-29 CN disclosed
EP-2066631-A1 PYRIDINE BORANE COMPLEXES BASF SE (DE) 2009-06-10 EP disclosed
WO-2008034886-A1 PYRIDINE BORANE COMPLEXES BASF SE (DE) 2008-03-27 WO disclosed