SCHEMBL4003060

SCHEMBL4003060

CC(C)(C)c1ccc(CN(C(=O)C(=O)O)c2ccc(Br)cc2C(F)(F)F)cc1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR9 P51686 1/20 0.42
SERPINE1 P05121 7/20 0.39
NR1H4 Q96RI1 1/20 0.38
PTGES O14684 2/20 0.37
ALOX5 P09917 2/20 0.37
ESRRG P62508 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
HDAC6 Q9UBN7 4/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC11 Q96DB2 3/20 0.35
STAT3 P40763 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1239528 0.88 CCR9 (0.38) CCR9NR1H4PTGESALOX5ESRRG
SCHEMBL4008718 0.84 PTPN1 (0.43) CCR9SERPINE1NR1H4PTGESALOX5
SCHEMBL4010103 0.81 SERPINE1 (0.48) SERPINE1NR1H4PTGESALOX5HDAC6
SCHEMBL1241613 0.80 SERPINE1 (0.49) SERPINE1NR1H4
SCHEMBL1241573 0.80 SERPINE1 (0.57) SERPINE1NR1H4PTGESALOX5
SCHEMBL4006485 0.80 SERPINE1 (0.45) SERPINE1NR1H4PTGESALOX5HDAC6
SCHEMBL4441053 0.78 NR1H4 (0.52) CCR9SERPINE1NR1H4PTGESALOX5
SCHEMBL4005059 0.77 NR1H4 (0.43) CCR9SERPINE1NR1H4PTGESALOX5
SCHEMBL1242713 0.75 SERPINE1 (0.58) SERPINE1NR1H4PTGESALOX5
SCHEMBL1241447 0.73 PTPN1 (0.41) CCR9NR1H4HDAC6HDAC8HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2072498-A1 N-PHENYLOXAMIDIC ACID DERIVATIVE Institute of Medicinal Molecular Design, Inc. (JP) 2009-06-24 EP disclosed