SCHEMBL4008718

SCHEMBL4008718

CC(C)(C)c1ccc(CN(C(=O)C(=O)O)c2ccc(Br)cc2OC(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.43
CCR9 P51686 1/20 0.42
SERPINE1 P05121 8/20 0.41
PTGER1 P34995 1/20 0.39
GCGR P47871 2/20 0.39
GIPR P48546 2/20 0.39
GLP1R P43220 1/20 0.39
NR1H4 Q96RI1 2/20 0.38
EPHX2 P34913 1/20 0.38
HRH4 Q9H3N8 2/20 0.37
HIF1A Q16665 1/20 0.37
EPAS1 Q99814 1/20 0.37
CACNA1H O95180 1/20 0.36
PTGES O14684 1/20 0.35
ALOX5 P09917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1241447 0.90 PTPN1 (0.41) PTPN1CCR9PTGER1GCGRGIPR
SCHEMBL1241436 0.85 SERPINE1 (0.56) SERPINE1GCGRGIPRGLP1RNR1H4
SCHEMBL4003060 0.84 CCR9 (0.42) CCR9SERPINE1NR1H4PTGESALOX5
SCHEMBL14635713 0.79 SERPINE1 (0.44) PTPN1SERPINE1PTGER1HRH4HIF1A
SCHEMBL1241445 0.79 SERPINE1 (0.52) PTPN1SERPINE1GCGRGIPRGLP1R
SCHEMBL1239797 0.78 SERPINE1 (0.46) SERPINE1GCGRGIPRGLP1RNR1H4
SCHEMBL1242219 0.77 SERPINE1 (0.54) SERPINE1GCGRGIPRGLP1RNR1H4
SCHEMBL1239503 0.76 SERPINE1 (0.56) SERPINE1GCGRGIPRGLP1RNR1H4
SCHEMBL1241573 0.76 SERPINE1 (0.57) SERPINE1GCGRGIPRGLP1RNR1H4
SCHEMBL1241454 0.76 SERPINE1 (0.55) SERPINE1GCGRGIPRGLP1RNR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2072498-A1 N-PHENYLOXAMIDIC ACID DERIVATIVE Institute of Medicinal Molecular Design, Inc. (JP) 2009-06-24 EP disclosed