SCHEMBL4005873

SCHEMBL4005873

CN(C=O)OC[C@@]1(Cc2cc(F)cc(NC(=O)Nc3cccnc3)c2)CCCNC1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
CHRNA7 P36544 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
LMNA P02545 2/20 0.37
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4010563 0.95 TAAR1 (0.42) CYP1A2CHRNA7TAAR1LMNAMEN1
SCHEMBL4012585 0.89 CHRNA7 (0.34) CHRNA7
SCHEMBL4011309 0.84 ROCK2 (0.33) CYP1A2MEN1KMT2A
SCHEMBL5072945 0.78 CHRNA7 (0.36) CHRNA7MAPT
SCHEMBL4006505 0.78 CHRNA7 (0.36) CHRNA7MAPT
SCHEMBL397837 0.77 TAAR1 (0.52) CYP1A2TAAR1LMNAMEN1ALDH1A1
SCHEMBL402340 0.75 TAAR1 (0.47) CYP1A2TAAR1LMNAMEN1ALDH1A1
SCHEMBL403106 0.72 CYP1A2 (0.49) CYP1A2TAAR1MEN1ALDH1A1KMT2A
SCHEMBL402800 0.72 CYP1A2 (0.51) CYP1A2TAAR1MEN1KMT2A
SCHEMBL400879 0.71 CYP1A2 (0.50) CYP1A2TAAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765327-A4 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS INC (US) 2009-06-17 EP claimed
EP-1765327-A2 COMPOUNDS, COMPOSITIONS AND METHODS Cytokinetics, Inc. (US) 2007-03-28 EP claimed
WO-2006009726-A2 SUBSTITUTED UREA DERIVATIVES FOR TREATING CARDIAC DISEASES CYTOKINETICS, INC. (US) 2006-01-26 WO claimed
EP-1765327-A4 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS INC (US) 2009-06-17 EP disclosed
EP-1765327-A2 COMPOUNDS, COMPOSITIONS AND METHODS Cytokinetics, Inc. (US) 2007-03-28 EP disclosed
WO-2006009726-A2 SUBSTITUTED UREA DERIVATIVES FOR TREATING CARDIAC DISEASES CYTOKINETICS, INC. (US) 2006-01-26 WO disclosed