SCHEMBL4009996

SCHEMBL4009996

CCCc1nc(C)n(-c2cccc(OC(C)C)c2)c(=O)c1Cc1cccc(-c2ccccc2)c1C#N

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 5/20 0.37
CD274 Q9NZQ7 2/20 0.37
CYP2C9 P11712 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
CCKBR P32239 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1892100 0.86 PPARG (0.39) S1PR1CYP2C9
SCHEMBL4016374 0.84 F10 (0.40) CD274SMN1; SMN2
SCHEMBL4013365 0.83 SMN1; SMN2 (0.40) CD274SMN1; SMN2
SCHEMBL4313277 0.79 CD274 (0.41) CD274
SCHEMBL1892524 0.78 AGTR1 (0.40)
SCHEMBL1885801 0.77 SLC33A1 (0.51)
SCHEMBL4450943 0.77 CYP3A4 (0.39) CD274CYP2C9CYP1A2CYP3A4MAPT
SCHEMBL1893662 0.76 PPARG (0.39) S1PR1CYP2C9
SCHEMBL1892613 0.75 PPARG (0.38) S1PR1CYP2C9
SCHEMBL1886447 0.75 PPARG (0.39) S1PR1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed