SCHEMBL4010154

SCHEMBL4010154

CCN(CC)CCOc1ccc(NC(=O)CNc2c(F)c(F)c(C)c(F)c2F)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.53
KDM4E B2RXH2 1/20 0.50
HTT P42858 1/20 0.43
HRH3 Q9Y5N1 2/20 0.42
RORC P51449 1/20 0.42
MAPT P10636 3/20 0.42
LMNA P02545 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
MCHR1 Q99705 3/20 0.41
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
MAOA P21397 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4015413 0.95 KDR (0.51) KDRKDM4EHTTHRH3RORC
SCHEMBL14209512 0.80 KDR (0.60) KDRKDM4EHTTHRH3RORC
SCHEMBL3865174 0.80 KDR (0.62) KDRKDM4EHTTHRH3RORC
SCHEMBL4011687 0.79 KDM4E (0.46) KDRKDM4EHTTRORCMAPT
SCHEMBL13811535 0.79 KDR (0.59) KDRKDM4EHTTHRH3RORC
Bromide SCHEMBL4014245 0.79 KDR (0.59) KDRKDM4EHTTHRH3RORC
SCHEMBL4007924 0.79 KDR (0.47) KDRKDM4EHTTHRH3MAPT
SCHEMBL4009187 0.79 KDR (0.49) KDRKDM4EHTTHRH3RORC
SCHEMBL4015144 0.78 BCHE (0.48) KDRKDM4EHTTRORCMAPT
SCHEMBL4014447 0.77 HRH3 (0.48) KDRKDM4EHTTHRH3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558567-B1 NOVEL AMIDE COMPOUNDS WITH MCH ANTAGONISTIC EFFECT AND MEDICAMENTS COMPRISING SAID COMPOUNDS BOEHRINGER INGELHEIM PHARMA (DE) 2009-06-24 EP claimed