SCHEMBL4010732

SCHEMBL4010732

CN(C)C1(c2ccccc2)CCC(c2cn(CCO)c3ccccc23)CC1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 12/20 0.43
OPRM1 P35372 8/20 0.43
CNR2 P34972 1/20 0.43
HRH2 P25021 4/20 0.40
OPRK1 P41145 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL735181 0.73 HTR6 (0.43) OPRL1OPRM1CNR2OPRK1
SCHEMBL733041 0.70 OPRL1 (0.48) OPRL1OPRM1OPRK1
SCHEMBL3144048 0.67 OPRL1 (0.62) OPRL1OPRM1OPRK1
SCHEMBL736413 0.67 OPRL1 (0.60) OPRL1OPRM1OPRK1
SCHEMBL27494196 0.67 HRH2 (0.45) HRH2
SCHEMBL733990 0.66 OPRM1 (0.47) OPRL1OPRM1OPRK1
SCHEMBL5166463 0.66 OPRL1 (0.61) OPRL1OPRM1
SCHEMBL13650541 0.66 OPRL1 (0.58) OPRL1OPRM1OPRK1
SCHEMBL27559062 0.65 HRH2 (0.59) CNR2HRH2
SCHEMBL5382074 0.65 OPRL1 (0.68) OPRL1OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044016-A2 4-HETEROARYL-SUBSTITUTED 1-AMINOCYCLOHEXANE-1-AND CYCLOHEXENE-1-DERIVATIVES HAVING EFFECTS ON THE OPIOD RECEPTOR SYSTEM Grünenthal GmbH (DE) 2009-04-08 EP disclosed
WO-2008009415-A2 4-HETEROARYL-SUBSTITUTED 1-AMINOCYCLOHEXANE-1- AND CYCLOHEXENE-1-DERIVATIVES HAVING EFFECTS ON THE OPIOD RECEPTOR SYSTEM Grünenthal GmbH (DE) 2008-01-24 WO disclosed