SCHEMBL4011571

SCHEMBL4011571

O=C(c1ccccc1)c1cncc(N2CC3CNC(C3)C2)c1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 6/20 0.55
CHRNA4 P43681 6/20 0.55
CHRNB4 P30926 15/20 0.55
CHRNA3 P32297 15/20 0.55
CHRNA7 P36544 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2961067 0.90 CHRNB4 (0.51) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL2955968 0.88 CHRNB4 (0.53) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL5996594 0.87 CHRNB4 (0.70) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL5987239 0.81 CHRNB2 (0.74) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL2961069 0.81 CHRNB2 (0.74) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL2954949 0.81 CHRNB2 (0.74) CHRNB2CHRNA4CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL2958574 0.80 CHRNB2 (0.72) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL4003627 0.79 CHRNB4 (0.73) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL4007434 0.79 CHRNB4 (0.73) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL2963531 0.78 CHRNB4 (0.48) CHRNB2CHRNA4CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081246-A2 BICYCLIC DIAMINES AS NICOTINIC RECEPTOR AGONISTS PFIZER INC. (US) 2009-07-02 WO claimed
WO-2009081246-A2 BICYCLIC DIAMINES AS NICOTINIC RECEPTOR AGONISTS PFIZER INC. (US) 2009-07-02 WO disclosed
WO-2009081246-A2 BICYCLIC DIAMINES AS NICOTINIC RECEPTOR AGONISTS PFIZER INC. (US) 2009-07-02 WO disclosed