SCHEMBL4012176

SCHEMBL4012176

Cc1cc(-c2cc(-c3ccccc3)cc(S(C)(=O)=O)c2Cl)c2cccc(C(F)(F)F)c2n1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 16/20 0.46
NR1H3 Q13133 14/20 0.46
RXRA P19793 2/20 0.39
ESR1 P03372 1/20 0.39
P2RX7 Q99572 1/20 0.38
RORC P51449 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27786952 0.89 NR1H2 (0.49) NR1H2NR1H3RXRAESR1
SCHEMBL27765362 0.80 CD38 (0.38) NR1H2NR1H3ESR1RORC
SCHEMBL4010226 0.78 NR1H2 (0.57) NR1H2NR1H3RXRA
SCHEMBL4012475 0.74 NR1H2 (0.58) NR1H2NR1H3RXRA
SCHEMBL27786951 0.74 NR1H2 (0.46) NR1H2NR1H3RXRA
SCHEMBL4017313 0.74 NR1H2 (0.70) NR1H2NR1H3RXRA
SCHEMBL27786950 0.73 CD38 (0.41) NR1H2NR1H3ESR1
SCHEMBL4010841 0.71 RORC (0.40) NR1H2NR1H3RXRAESR1RORC
SCHEMBL4011954 0.70 NR1H2 (0.73) NR1H2NR1H3RXRA
SCHEMBL4017110 0.69 NR1H2 (0.57) NR1H2NR1H3RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN claimed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed