SCHEMBL4010841

SCHEMBL4010841

Cc1cc(-c2cc(OS(=O)(=O)C(F)(F)F)ccc2Cl)c2cccc(C(F)(F)F)c2n1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RORC P51449 10/20 0.40
NR1H2 P55055 8/20 0.36
NR1H3 Q13133 8/20 0.36
RXRA P19793 1/20 0.36
ESR1 P03372 1/20 0.35
BDKRB2 P30411 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4014835 0.88 NR1H2 (0.39) RORCNR1H2NR1H3RXRAESR1
SCHEMBL4012142 0.85 ENPP1 (0.44) RORC
SCHEMBL4017110 0.83 NR1H2 (0.57) NR1H2NR1H3RXRA
SCHEMBL4019268 0.81 NR1H2 (0.59) NR1H2NR1H3RXRA
SCHEMBL4018710 0.80 NR1H2 (0.55) NR1H2NR1H3RXRA
SCHEMBL4014198 0.79 NR1H3 (0.47) RORCNR1H2NR1H3RXRA
SCHEMBL3508705 0.79 LPAR1 (0.39) NR1H2NR1H3RXRA
SCHEMBL4013024 0.79 NR1H2 (0.56) NR1H2NR1H3RXRA
SCHEMBL4012143 0.78 ESR1 (0.40) RORCESR1BDKRB2
SCHEMBL4018305 0.78 NR1H2 (0.45) RORCNR1H2NR1H3RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed