SCHEMBL4012184

SCHEMBL4012184

COc1cccc(-c2cc(C)nc3c(C(F)(F)F)cccc23)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 5/20 0.46
NR1H3 Q13133 4/20 0.46
RXRA P19793 1/20 0.46
PGR P06401 1/20 0.45
AR P10275 1/20 0.45
AKR1C4 P17516 1/20 0.45
AKR1C3 P42330 1/20 0.45
AKR1C2 P52895 1/20 0.45
AKR1C1 Q04828 1/20 0.45
ESR1 P03372 1/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4015511 0.82 ENPP1 (0.40) ESR1NPC1RAB9ATSHRHTT
SCHEMBL4014169 0.82 PIK3CD (0.46) NR1H2NR1H3ARESR1ALDH1A1
SCHEMBL4012142 0.81 ENPP1 (0.44) RAB9ASMN1; SMN2TSHRHTT
SCHEMBL4011954 0.81 NR1H2 (0.73) NR1H2NR1H3RXRA
SCHEMBL3506710 0.80 ADORA2A (0.48) NR1H2NR1H3PGRARESR1
SCHEMBL4011974 0.79 NR1H2 (0.66) NR1H2NR1H3RXRA
SCHEMBL4012015 0.79 NR1H2 (0.74) NR1H2NR1H3RXRA
SCHEMBL4013511 0.77 NR1H2 (0.67) NR1H2NR1H3RXRA
SCHEMBL4010727 0.76 NR1H3 (0.58) NR1H2NR1H3RXRA
SCHEMBL4017313 0.76 NR1H2 (0.70) NR1H2NR1H3RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed