SCHEMBL4014169

SCHEMBL4014169

Cc1cc(-c2cccc(O)c2)c2cccc(C(F)(F)F)c2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.46
ESR1 P03372 2/20 0.42
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HSD17B1 P14061 2/20 0.41
HSD17B2 P37059 2/20 0.41
NR1H2 P55055 4/20 0.41
NR1H3 Q13133 4/20 0.41
AR P10275 1/20 0.41
ENPP1 P22413 1/20 0.40
CD38 P28907 3/20 0.39
CYP3A4 P08684 2/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
CCNE2 O96020 1/20 0.39
CDK4 P11802 1/20 0.39
CCND1 P24385 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
MET P08581 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4012780 0.82 CD38 (0.41) ESR1GAAMAPTHSD17B1HSD17B2
SCHEMBL4012184 0.82 NR1H2 (0.46) ESR1NR1H2NR1H3ARCYP3A4
SCHEMBL4013817 0.81 NR4A2 (0.54) PIK3CDGAAMAPTHSD17B1HSD17B2
SCHEMBL4012143 0.81 ESR1 (0.40) ESR1GAAMAPTHSD17B1HSD17B2
SCHEMBL1125582 0.80 NR1H2 (0.62) PIK3CDHSD17B1HSD17B2NR1H2NR1H3
SCHEMBL3507496 0.78 ESR1 (0.42) PIK3CDESR1GAAHSD17B1HSD17B2
SCHEMBL3278103 0.78 PIK3CD (0.43) PIK3CDESR1HSD17B1HSD17B2NR1H2
SCHEMBL9494183 0.78 CD38 (0.44) ESR1GAAMAPTHSD17B1HSD17B2
SCHEMBL4017313 0.78 NR1H2 (0.70) NR1H2NR1H3
SCHEMBL6479303 0.75 KDM4E (0.59) ESR1GAAMAPTCD38CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed